Japanese Society for Process Chemistry
 
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⇒Paticipants of Symposium
⇒Lecture & Poster Presentation
⇒JSPC Award for Excellence
⇒2010`2012
Ë2005`2009
Ë2002`2004
 
 



2009

JSPC 2009 Winter Symposium

December 4, 2009
Kyoto Terrsa
Organizer: Hiroshi Oshima (Osaka Prefecture Univ.), Toru Sugaya(Daiichi Fine Chemical)

<Invited Lectures>

  1. Industrial Process Development by Enzymation
    Keiji Sakamoto
    (Product Development Department, Daiichi Fine Chemical Co., Ltd.)
    Chair : Hitoshi Arai (Kyowa Hakko Kirin)

  2. How to make Dry Powder by Spray Drying-Process and Particle Design
    Masaaki Okawara*, Takashi Itou, Tosiyuki Tanaka
    (Development Dept., Ohkawara Kakohki Co., Ltd.)
    Chair : Koji Kagara (Ohara)

  3. Synthetic Organic Reactions with Indobenzenes as Organocatalysts
    Masahito Ochiai
    (Graduate School of Pharmaceutical Sciences, University of Tokushima)
    Chair : Toshiro Konoike (Shionogi)

  4. The Metalated Flatland Conduit to New Synthetic Aromatics and Heteroaromatic Chemistry
    Victor Snieckus
    (Department of Chemistry, Queen's University)
    Chair : Kiyoshi Tomioka (Kyoto Univ.)

<JSPC Award for Excellence 2009 Lecture>  Chair: Takahiko Akiyama (Gakushuin Univ.)

  1. Direct Oxidative Conversion of Alcohols, Amines, and Alkyl halides into Nitriles with Molecular Iodine and 1,3-Diiodo-5,5-dimethylhydantoin in aq. Ammonia. Shinpei Iida, Ryosuke Ohmura, Hideo Togo*
    (Graduate School of Science, Chiba University, Japan)

  2. Optimization of drying process in scale-up manufacturing for Erythromycin A derivative. Kaichiro Koyama*, Hitoshi Shimizu, Shinichi Ebihara
    (synthetic Technology Research Dept., Chugai Pharmaceutical & Co., Ltd., Japan)

  3. An Efficient Synthesis of Chiral Alcohols via Catalytic Hydrogen Reduction of Esters.
    Osamu Ogata*, Yasunori Ino, Wataru Kuriyama, Takaji Matsumoto
    (Corporate research & Development Division, Takasago International Corporation, Japan)

  4. Development of very mild and highly selective deprotection method of methylene acetals.
    Hiromichi Fujioka, Kento Senami*, Ozora Kubo, Yutaka Minamitsuji, Tomohiro Maegawa
    (Graduate School of Pharmaceutical Sciences, Osaka University, Japan)

 
JSPC 2009 Summer Symposium

July 16-17, 2009
Tower Hall Funabori
Organizer: Takahiko Akiyama (Gakushuin Univ.) , Akihiko Miyadera (Daiichi-Sankyo)

<Invited Lectures>

  1. Time-saving, Cost-effective, Totally Efficient Condensations Directed for Process Chemistry
    Yoo Tanabe
    (Department of Chemistry, School of Science and Technology, Kwansai Gakuin University)
    Chair : Toshiro Konoike (Shionogi)

  2. Complete Switch of Product Selectivity in Asymmetric Reaction with Two Chiral Organocatalysts from a Common Chiral Source
    Keiji Nakayama
    (Process Technology Research Laboratories, Daiichi-Sankyo Co., LTD.)
    Chair : Takahiko Akiyama (Gakushuin Univ.)

  3. Selective Cross-Coupling Reactions Catalyzed by Iron
    Masaharu Nakamura
    (International research Center for Elements Science, Institute for Chemical Research, Kyoto University)
    Chair : Hironao Sajiki (Gifu Pharmaceutical Univ.)

  4. New Possibility for Design of Catalysis
    Tohru Yamada
    (Department of Chemistry, Keio University)
    Chair : Masahiro Oshima (Tanabe Mitsubishi)

  5. Novel Recycling System Utilizing New Polymer-Gel Catalysts in Organic Synthesis
    Shiro Ikegami
    (Teikyo University)
    Chair : Takayuki Shioiri (Meijo Univ.)

  6. Ozonolysis in Manufacturing Process
    Haruo Koike
    (Nichia Pharmaceutical Industries LTD.)
    Chair : Kin-ichi Tadano (Keio Univ.)

  7. Process Development of Chiral cis-1-Aminoindan-2-ol in Industrial Scale
    Yoshio Igarashi
    (Tama Kagaku Kogyo Co. Ltd.)
    Chair : Koji Kagara (Ohara)

  8. Efficient Synthesis of Maxacalcitol, the Vitamin D3 Analogue Exhibiting Low Calcemic Activity
    Hitoshi Shimizu
    (Synthetic Technology Research Department, Chugai Pharmaceutical Co., Ltd.)
    Chair : Takumi Tanaka (Wako)

  9. Process Research on a Novel Anticancer Drug E7389 (Eribulin mesylate)
    Katsuya Tagami
    (Kashima Process Research, API Research Laboratories, Eisai Co., Ltd.)
    Chair : Ryuji Mukuta (Astellas)

  10. Mechanism and Control of Polymorph and Quasi-Polimorph Appearance in Crysrallization of Organic Compounds
    Hiroshi Ooshima
    (Guraduate School of Engineering, Osaka City University)
    Chair : Shigeru Soda (Eisai)

  11. About recent solvent recycling -Mainly Japanese, China in the center of the topic-
    Yasuhito Kawase
    (Nippon Refine Co., Ltd.)
    Chair : Toyonori Takebayashi (Daiichi-Sankyo Chemical Pharma)
¡JSPC Award for Excellence 2009 >>

¡
Grant-in-Aid for Scientific Research on Priority Areas
Advanced Molecular Transformations of Carbon Resources Symposium

June 1-2, 2009
Kyoto Terrsa

<Invited Lectures>

  • Keiji Maruoka (Kyoto Univ.)
  • Kei Manabe (Univ. of Shizuoka)
  • Masaya Sawamura (Hokkaido Univ.)
  • Akira Yanagisawa (Chiba Univ.)
  • Yutaka Ukaji (Kanazawa Univ.)
  • Makoto Shimizu (Mie Univ.)
  • Masahiko Hayashi (Kobe Univ.)
  • Takahiko Akiyama (Gakushuin Univ.)
  • Yoo Tanabe (Kwansai Gakuin Univ.)
  • Makoto Nakajima (Kumamoto Univ.)
  • Ken Kamikawa (Osaka Prefecture Univ.)
  • Isamu shiina (Tokyo Univ. of Science)
  • Fumitoshi Kakiuchi (Keio Univ.)
  • Kyoko Nozaki (Univ. of Tokyo)
  • Ilhyong RYU (Osaka Prefecture Univ.)
  • Nobuaki Kambe (Osaka Univ.)
  • Michinori Suginome (Kyoto Univ.)
  • Susumu Saito (Nagoya Univ.)
  • Tsumoru Kakiuchi (Nara Institute of Science and Technology)
  • Yasutaka Ishii (Kansai Univ.), Yasusi Obora (Kansai Univ.)
  • Takahiro Nishimura (Kyoto Univ.)
  • Teruyuki Kondo (Kyoto Univ.)
  • Kazuhiko Takai (Okayama Univ.)
  • Tsugio Kitamura (Saga Univ.)
  • Shinobu Ito (Osaka Univ.)
  • Junzo Odera (Okayama Univ.)
  • Kiyoshi Tomioka (Kyoto Univ.)
  • Masami Kamigaito (Nagoya Univ.)
  • Atsuki Mori (Koube Univ.)
  • Koichi Ohe (Kyoto Univ.)
  • Atsushi Kawauchi (hiroshima Univ.)

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2008

 
The Pharmaceutical Society of Japan (PSJ) 129th SymposiumF Impact of Pharmaceutical Process Chemistry

March 28, 2009
Kyoto International Conference Center
Organizer: Yasumaru Hatanaka (Toyama Univ.), Yozo Todo (Toyama Chemical), Takayuki Shioiri (Meijo Univ.)

<Invited Lectures>

  1. Yozo Todo (Toyama Chemical Co., Ltd.)

  2. Masaru Mitsuda (Kaneka)

  3. Masayuki Yabuta (Asubio Pharma Co. Ltd)

  4. Masahiko Kinugawa (kyowa Hakko Kirin)

 
JSPC 2008 Winter Symposium

December 1, 2008
Tower Hall Funabori
Organizer: Takumi Tanaka (Wako), Takahiko Akiyama (Gakushuin Univ.)

<Invited Lectures>

  1. Synthetic Studies on Azacycles Based on Process Chemistry for New Drug Candidates
    Hideya Mizufune
    (Chemical Development Laboratories, CMC Center, Pharmaceutical Prodection Division, Takeda Pharmaceutical Company Limited)
    Chair : Tomoyuki Onishi (Ajinomoto)

  2. Research for Establishing Practical CIDT Process
    Yoshihiko Tarai*, Kenichi Toyama, Tadashi Shirasaka, Hiroshi Iwamura
    (Process Chemistry Research Development, CMC Research Center, Mitsubishi Tanabe Pharma Corporation)
    Chair : Nobuhiro Ito (Wako)

  3. Advances in Process Chemistry of Cross-Coupling Reactions
    Norio Miyaura
    (Graduate School of Engineering, Hokkaido University)
    Chair : Kin-ichi Tadano (Keio Univ.)

  4. Development of Separation Process
    Masakuni Matsuoka
    (Tokyo University of Agriculture and Technology)
    Chair : Takayuki Shioiri (President of JSPC)

ƒJSPC Award for Excellence 2008 Lecture„ Chair : Hironao Sajiki (Gifu Pharmaceutical Univ.)

  1. A Practical Synthesis of the PDE4 inhibitor KW-4490.
    Arata Yanagisawa*, Koichiro Nishimura ,Tetsuya Nezu, Kyoji Ando, Ayako Maki, Eiichiro Imai, Shin-ichiro Mohri
    (Kyowa Hakko Kogyo, Japan)

  2. An Efficient Synthesis of the PKCb Inhibitor JTT-010 Using a Novel Cyclopropane Ring-Opening Reaction with Indole
    Takashi Inaba*, Masahiro Tanaka, Minoru Ubukata, Takafumi Matsuo, Katsutaka Yasue, Katsuya Matsumoto, Yasuyuki Kajimoto, Takashi Ogo
    (Japan Tobacco Inc.,Japan)

  3. Development of Protecting Group Free Catalytic O-Selective Acylation of Aminoalcohols
    Takashi Ohshima*, Takanori Iwasaki, Yusuke Maegawa, Yukiko Hayashi, Kazushi Mashima
    (Osaka University, Japan)

  4. Dramatic Kinetic Resolution of Primary Amines by Lipase-Palladium Cocatalysis
    ›Kiwon Han, Yoon Kyung, Cheolwoo Kim, Jaiwook Park, Mahn-Joo Kim
    (POSTEC, Korea)

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¡
The First International Symposium on Process Chemistry [ISPC 08]

Kyoto International Conference Center
July 28 (Mon) - 30 (Wed), 2008
Chair Takayuki Shioiri (Meijo Univ.)

<Keynote Lecture>

@@@@@yJuly 29 (Tue)z

  1. From Milligrams to Tons: The Importance of Synthesis & Process Research in the Development of New Drugs
    Martin Karpf (F. Hoffmann-La Roche, Switzerland)
    Chair: Toshiro Konoike (Shionogi, Japan)

  2. Streamlining Synthesis via C-H Oxidation
    M. Christina White (Univ. of Illinois, Urbana-Champaign, USA)
    Chair: Hironao Sajiki (Gifu Pharm. Univ., Japan)

  3. Design of Dynamic Salt Catalysts Based on Acid-Base Combination Chemistry
    Kazuaki Ishihara (Nagoya Univ., Japan)
    Chair: Yoo Tanabe (Kwansei Gakuin Univ., Japan)

  4. Enzymo-Metallic Dynamic Kinetic Resolution as a New Tool for Chiral Synthesis
    Mahn-Joo Kim (Pohang Univ. of Sci. & Tec., Korea)
    Chair: Kenji Inoue (Kaneka, Japan)

  5. Matching Chemistry with Chemical Engineering for Optimum Design and Performance of Pharmaceutical Processing
    Aniruddha B. Pandit (Univ. of Mumbai, India)
    Chair: Koji Kagara (Ohara, Japan)

  6. Boron Reagents in Process Chemistry: Excellent Tools for Selective Reductions
    Karl Matos (BASF Corporation, USA)
    Chair: Yoshiharu Iwabuchi (Tohoku Univ., Japan)

  7. Asymmetric Oxidation with Hydrogen Peroxide, an Effective and Versatile Oxidant
    Tsutomu Katsuki (Kyushu Univ., Japan)
    Chair: Masakatsu Shibasaki (Univ. of Tokyo, Japan)

    yJuly 30 (Wed)z

  8. Process Development of HIV Integrase Inhibitor S-1360
    Toshiro Konoike (Shionogi, Japan)
    Chair: Ichiro Shinkai (Beta Chem, Japan)

  9. An Entirely New Methodology for Synthesizing Perfluorinated Compounds
    Takashi Okazoe (Asahi Glass, Japan)
    Chair: Noritada Matsuo (Sumitomo Chem., Japan)

  10. New Methods for the Functionalization of Aromatic Compounds
    Keith Fagnou (Univ. of Ottawa, Canada)
    Chair: Yujiro Hayashi (Tokyo Univ. of Science, Japan)

  11. Byproduct-Free C-C Bond Formation via Catalytic Hydrogenation and Transfer Hydrogenation
    Michael J. Krische (Univ. of Texas at Austin, USA)
    Chair: Takahiko Akiyama (Gakushuin Univ., Japan)

  12. Commercialization of a Sodium Hydride Mediated Arylation Process
    Mark Butchko (Eli Lilly, USA)
    Chair: Norio Hashimoto (Astellas, Japan)

  13. Design Space for Drug Substance - the Approach used for Vandetanib
    David Haywood (AstraZeneca, UK)
    Chair: Kunisuke Izawa (Ajinomoto, Japan)

<JSPC Award for Excellence 2007 Lecture>@Chair: Takumi Tanaka (Wako, Japan)

  1. Process development of a key building block for anti-AIDS drugs by proline catalyzed enatio-selective direct cross aldol reaction
    Tetsuya Ikemoto*, Yosuke Watanabe, Junichi Tomokawa, Takehiko Kawakami, Yasuo Uekita, Isao Kurimoto (Sumitomo Chem., Japan)

  2. Catalytic Reduction of Carboxamides by Hydrosilanes
    Hideo Nagashima*, Hidehiro Sasakuma, Nariaki Harada, Hironori Tsutsumi, Yukihiro Motoyama (Kyushu Univ., Japan)

  3. Development of One-pot Synthesis of New Antiarthritic Drug Candidate S-2474 with High E-Selectivity
    Takemasa Hida*, Katsuo Oda, Hideo Nogusa, Toshiaki Masui (Shionogi, Japan)

URL:@http://www.chemicaldaily.co.jp/ent/process_g/index.html

This symposium came to an end with great success by 996 people participating. (57 people in foreign countries) Thank you very much for a lot of cooperation of participant.
¡JSPC Award for Excellence 2008>>

2007

 
Grant-in-Aid for Scientific Research on Priority Areas
Advanced Molecular Transformations of Carbon Resources Joint Symposium

December 6-7, 2007
Kyoto Terrsa
Organizer: Toshiaki Mase (Banyu), Kiyoshi Tomioka (Kyoto Univ.)

ƒInvited Lectures„

y12/6z

@Chair : Kyoko Nozaki

  • Efficient Syntheses of Multisubstituted Cyclic Molecules Initiated by Ynolates
    Mitsuru Shindo
    iInstitute for Materials Chemistry and Engineering, Kyusyu Universityj

  • New Catalytic Transformations for Propargylic Amines
    Hiroyuki Nakamura
    iDepartment of Chemistry, Faculty of Science, Gakushuin Universityj

@Chair : Yasutaka Ishii

  • Selective Oxidation Reactions Cataluzed by Finely-tuned Active Sites on Polyoxometalates
    Shiro Hikichi
    (Faculty of Engineering, Department of Material and Life Chemistry, Kanagawa University)

  • Towards Enantioselective Nucleophilic Trifluoromethylation Reactions
    Norio Shibata
    (Department of Applied Chemistry, Nagoya Institute of Technology)

@Chair : Junzo Odeta

  • Versatile Molecular Transformations Using Vanadium Redox Catalysts
    Toshikazu Hirao
    (Graduate School of Engineering, Osaka University)

  • Construction of p-Conjugated Heteroaromatic Compounds via Palladium-catalyzed CH Arylation
    Atsunori Mori
    iGraduate School of Engineering, Kobe Universityj

@Chair : Keiji Maruoka

  • Chiral BrØnsted Acid-Catalyzed Enantioselective Synthesis of Nitrogen-Containing Compounds
    Takahiko Akiyama
    iFaculty of Science, Gakushuin Universityj

  • Catalyst-free Efficient Reactions in Dimethyl Sulfoxide
    Takeshi Oriyama
    (Faculty of Science, Ibaraki University)

Chair : Tomohiko Owada

  • Development of Copper(I) Catalysis Based on Ligand-Control Concept
    Masaya Sawamura
    (Faculyu of Science, Hokkaido University)

  • One-Pot Selective Plural Carbon-Bond Formation though Oganic Electron Transfer Reactions
    Ikuzo Nishiguchi
    (Nagaoka University of Technology, Department of Chemistry)

  • A New Catalytic System: Development of Hg(OTf)2-Catalyzed Reactions
    Mugio Nishizawa
    (Faculty of Pharmaceutical Sciences, Tokushima Bunri University)

@Chair : Toshiaki Mase

  • uPreparation of CCR5 Drug Canditatev
    Nobuyoshi Yasuda
    (Merck Research Labs, Process Research)

  • Tetsu Yamakawa
    (Sagami Chemical Research Institute)

  • Protease-targeted Drug Discovery
    Genji Iwasaki
     (Novartis Institutes for BioMedical Research, Tsukuba)

y12/7z

@Chair : Toshiro Konoike

  • Mokecular Conversion of Carbon Monoxide via Radical/Ionic Cascade Reactions
    Ilhyong Ryu
    (Graduate School of Schience, Osaka Prefecture University)

  • Development of Advanced Molecular Transformations Utilizing Carbon-Carbon Bond Claevage
    Takahiro Nishimura
    (Graduate School of Science, Kyoto University)

  • Green Oxidation with Aqueous Hydrogen Peroxide
    Kazuhiko Sato
    (National Institute of Advanced Science and Technology (AIST))

  • Design and Application of Chiral Bifunctional Organocatalysts
    Keiji Maruyama
    (Graduate School of Science, Kyoto University)

Chair : Yoo Tanabe

  • uDiisobutylaluminium2,6-Di-tert-butyl-4-methylphenoxide. Novel Stereoselective Reducing Agent for Prostaglandin Synthesis
    Hisao Nakai
    (Medicinal Chemistry Research Laboratories, Research Headquaters, Ono Pharmaceutical Co., Ltd.)
    Development of A Novel Synthetic Method for RNA Oligomers: The Challenge of A Very Long RNA Oligomer
    Tadaaki Ohgi
    (Discovery Research Laboratories in Tsukuba, Nippon Shinyaku Co., Ltd)

  • Biotransformation-Induced New Possibility of Synthtic Route Design
    Manabu Katsurada
    (Biotechnology Laboratory, Mitsubishi Chemical Group Science and Technology Research Center, Inc.
    Bio& Chemical Process Discovery Laboratory, API Corporation)

  • Process Development of Anti-VLA-4 Drug, TRK-720
    Kazuharu Suyama*, Yuji Sugawara, Takami Kannno, Masayuki Maeda, Motohiro Shiraki, Kuniaki Kawamura, Katsuhiko Iseki
    (Pharmaceutical Research Laboratories, Toray Industries, Inc.)

  • Initial Process Reasearch for Ant^allergy Agents
    Keiji Nakayama
    (Process Technology Research Laboratories, Daiichi-Sankyo Co., LTD.)

 
JSPC 2007 Summer Symposium

August 2-3, 2007
Tower Hall Funabori
Organizer: Kuniaki Tatsuta (Waseda Univ.), Ryuji Mukuta (Astellas)

<Invited Lectures>

  1. Asymmetric Aldol Reaction Using Organocatalyst in the Presence of Water
    Yujiro Hayashi
    (Department of Industrial Chemistry, Faculty of Engineering, Tokyo University of Science)
    Chair: Hironao Sajiki (Gifu Pharmaceutical Univ.)

  2. Asymmetric Synthesis of Chiral Compounds Using Bifunctional Thioureas
    Yoshiji Takemoto
    (Graduate School of Pharmaceutical Sciences, Kyoto University)
    Chair: Akihiko Miyadera (Daiichi-Sankyo)

  3. Chiral BrØnsted Acid-Catalyzed Asymmetric Reactions
    Takahiko Akiyama
    (Department of Chemistry, Gakushuin University)
    Chair: Osamu Onomura (Nagasaki Univ.)

  4. Guanidine Chemistry: Discloure of its Potential Functionality
    Tsutomu Ishikawa
    (Graduate School of Pharmaceutical Sciences, Chiba University)
    Chair: Shunsuke Goto (Astellas)

  5. Development of Novel Process for Pharmaceutical Intermediated relevant to Amino Acid
    Kunisuke Izawa
    (AminoScience Laboratories, Ajinomoto Co., Inc.)
    Chair: Kenji Inoue (Kaneka)

  6. The Emerging Face of Indian Pharma Industry
    H.Garg
    (Senior Advisor, Asia, Oceania and Middle East Buisiness Headquaters Eisai Co., Ltd.)
    Chair: Toshiaki Mase (Banyu)

  7. Process Development of Optically Active β-Hydroxy-α-Amino Acid
    -Practical Application of anti-Serective Asymmetric Hydrogenation-
    Hideaki Kobayashi
    (Technical Developnment Division, Onoda Plant, Nissan Chemical Industries, Ltd.)
    Chair: Satoru Kuraoka (Tanabe)

  8. Case Study on Trouble in Practical Pilot Plant Productation
    -Manufacturing View-
    Toshiaki Masui
    (Industrial Technology Laboratories, Clinical Manufacturing Unit, Shionogi & Co., Ltd.)
    Chair: Takumi Tanaka (Wako)

  9. Two Complexity Phenomena in Chemistry Caused by Symmetry-Breaking
    Rui Tamura
    (Graduate School of Human and Environmental Studies, Kyoto University)
    Chair: Koji Machiya (Astellas)

  10. Solid-Liquid Separation by a Centrifuguge in Batch Crystallization Process
    Kunitoshi Takahashi
    (Utajima Pilot Production Dept./ Sumitomo Chemical Co., Ltd.)
    Chair: Toshiro Konoike (Shionogi)

  11. Measuremrnt of Drying Rates and Selectivity during Vaccumm Dryingof Pharmaceuticals and Analysis of The Mass Transfer Mechanism in a Layer of Crystalline Particles
    Masamichi Yoshida
    (Toyama University)
    Chair: Koji Kagara (Ohara)

@¡JSPC Award for Excellence 2007>>

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2006

 
JSPC 2006 Winter Symposium

Decemner 11, 2006
Tower Hall Funabori

<Invited Lectures>

  1. Yutaka Kameyama (Otsuka Fine Chemical)

  2. Hiromu Kawamura (Asahikasei Chemical Corporation)

  3. Takashi Isoda

  4. Yoshimitsu Nagao (Tokushima University)

<JSPC Award for Excellence 2006 Lecture> Chair : Akio Kayano (Eisai)

  1. Interesting characteristics and their control of polymorphs of bradykinin antagonist FR173657
    Ariyoshi Kubota, Koji Mukai, Shunsuke Goto, and Hironobu Yasuda
    (Astellas Pharma)

  2. Manufacturing process development of tricyclic triazolobenzazepine derivative
    Yumiko Okada, Shohei Yasuda, Jun Irie, Masaaki Takahashi, and Hitoshi Yamaguchi
    (Meiji Seika)

  3. Development of 1-methyl-AZADO: a highly efficient organocatalyst for oxidation of alcohols
    Yoshiharu Iwabuchi, Masatoshi Shibuya, Masaki Tomizawa, Takamune Hattori, and Takahisa Satoh
    (Tohoku Univ.)

 
JSPC 2006 Summer Symposium
(5th Symposium)

July 20-21, 2006
Kyoto Terrsa
Organizer: Yoo Tanabe (Kwansai Gakuin Univ.), Toshiro Konoike (Shionogi)

<Invited Lectures>

  1. Development of Industrial Process of Household Pyrethroid Insecticide
    Hiroshi Yamachika
    (Sumitomo Chemical Co., Ltd.)
    Chair: Yuzuru Saito (Takeda)

  2. Some Progress of Organic Synthesis of Pharmaceuticals in China
    W..Zhang
    (School of Chemistry and Chemical Engineering, Shanghai Jiao Tong University)
    Chair: Kazuo Shiraki (Wako)

  3. Process Development of Micafungin, a Novel Lipopeputide Antifungal Agent
    Atsushi Ohigashi
    (Process Chemistry Labs., Astellas Pharma Inc.)
    Chair: Hidetsura Cho (Japan Tabacco)

  4. Design of Chiral Organocatalysts for Practical Asymmetric Synthesis of Useful Amino Acid
    Keiji Maruoka
    (Dept. of Chem., Grad., of Sci., Kyoto University)
    Chair: Yoo Tanabe (Kwansai Gakuin Univ.)

  5. The Future Road to Process Chemistry
    Tetsuo Hiraoka
    (Sankyo Organic Chemicals Co., Ltd)
    Chair: Kiyoshi Tomioka (Kyoto Univ.)

  6. Process Research for API by autometic synthesis devices
    Hirofumi Kuroda*, Yoshihiko Hisatake, Akio Kayano, Kimihiro Matuo, Taiju Nakamura
    (Process Research Laboratories, Eisai & Co., Ltd.)
    Chair: Naoyuki Kishi (Sankyo)

  7. Application of Whole-Cll Biocatalysts in the Manufacture of Fine Chemicals
    Micheal Schwarn
    (Degussa AG, R&D Exclusive Synthesis)
    Chair: Hironao Sajiki (Gifu Pharmaceutical Univ.)

  8. New Possibilities Using Water as a Solvent in Organic Synthesis
    Shu Kobayashi
    (Graduate School of Pharmaceutical Sciences, The University of Tokyo)
    Chair: Takahiko Akiyama (Gakushuin Univ.)

  9. Practical Monohydrolysis of Symmetric Diesters
    Satomi Niwayama
    (Department of Chemistry and Biochemistry, Texas Tech University)
    Chair: Takayuki Shioiri (President of JSPC)

  10. Intellecture Property Management for Globalization of Drug Manufacturing
    Hirotsugu Takayama
    (Intellectual Property Dept., Shionogi & Co., Ltd.)
    Chair: Ryuji Mukuta (Astellas)

  11. Frontier of Pharmaceutical Quality Control: PAT on API
    Tatsuzo Ukita
    (CMC Research Laboratories, Pharmaceutical Development Dept., Tanabe Seiyaku Co., Ltd)
    Chair: Toshihiko Naito (Eisai)
¡JSPC Award for Excellence 2006>>

2005

¡
The Pharmaceutical Society of Japan (PSJ)132nd SymposiumF Enjoy the Process Chemistry

March 30, 2006
Sendai International Center
Organizer: Kozo Shishido (Tokushima Univ.), Shinji Aki (Otuka)

<Invited Lectures>

  1. Masato Matsugi (Meijo Univ.)

  2. Tomomi Ikemoto (Takeda)

  3. Hiroo Matsumoto (Nissan Chemical)

  4. Masaya Ikunaka (Nagase)

  5. Hiroki Ishibashi (Mitsui Chemical)


¡
JSPC 2005 Winter Symposium

December 8, 2005
Osaka Cent. Public Hall

<Invited Lectures>

  1. Two Case Studies on Process Development with Resolution vvis Diastereometric Salt Formation: their Chronological and Multifaceted Description to Identify the Real Competitiveness
    Masaya Ikunaka
    (Research & Development Center, Nagase & Co., Ltd.)
    Chair: Yuzuru Saito (Takeda)

  2. Synthetic Studies on the Medium-Sized Ring Lactones by Means of Rapid Lactonization Using Substituted Benzoic Anhydrides
    Isamu Shiina
    (Department of Applied Chemistry, Faculty of Science, Tyokyo University of Science)
    Chair: Yoo Tanabe (Kwansai Gakuin Univ.)

  3. Takanori Ushio1, Hidenori Miura1, Keiko Nagai1, Rui Tamura2
    (1Taiho Pharmaceutical Co., Ltd, 2Kyoto University)
    Chair: Tatsuzo Ukita (Tanabe)

  4. Development on New Drug and Crystal Polymorph
    Mitsuhisa Yamano
    (Chemical Development Laboratories, Takada Pharmaceutical Company Limited)
    Chair: Shunsuke Goto (Astellas)

<JSPC Award for Excellence 2005 Lecture>@Chair: Sakae Kobayashi (Wako)

  1. Practical process developments of KRP-103 for treatment of urinary incontinence
    Shintaro Kanazawa, Ichiro Araya
    (Research Center, Kyorin Pharmaceutical Co., Ltd.)

  2. Process development of BO-653 for large scale production
    Masahiro Nagase, Mitsuhiro Kurita, Takemi Tanokura, Motoki Shimizu, Yoshiaki Kato, Kunio Tamura, Hirohito Shimizu, Masahiro Kato
    (Syntthetic Technology Research Dept., Chugai Pharmaceutical Co., Ltd.)

  3. Lipase-Catalyzed Domino Synthesis: Kinetic Resolution of Racemic Alchols Followed by Intermolecular Cyclyzation
    Shuji Akai1, Kouichi Tanimoto2, Yukiko Kanao2, Sohei Omura2, Yasuyuki Kita2
    (1School of Pharmaceutical Sciences, University of Shizuoka, 2Graduate School of Pharmaceutical Sciences, Osaka University)

 
JSPC 2005 Summer Symposium

July 28-29, 2005
Tower Hall Funabori
Organizer: Takayuki Shioiri (Meijo Univ.), Shigeru Soda (Eisai)

<Invited Lectures>

  1. Process Development of an Angiotensin II Reseptor Antagonist
    Iwao Chujo
    (Sakai Research Laboratories, Kyowa Hakko Kyogyo, Co., Ltd.)
    Chair: Yoo Tanabe (Kwansai Gakuin Univ.)

  2. Development of New Asymmetric Catalyses for the Efficient Syntheses of α-Amino Acid Containing Natural Products
    Takashi Ohshima1,2, Tomoyuki Shibuguchi2, Hisashi Mihara2, Akihiro Okuda2, Yuhei Fukuta2, Masakatsu Shibasaki2
    (1Department of Chemistry, Graduate School of Engineering Science, Osaka University,
    2Graduate School of Pharmaceutical Sciences, The University of Tokyo)
    Chair: Sakae Kobayashi (Wako)

  3. Process Development of L-DOPA as Anti-Parkinson Drug
    Mitsusori Hashimoto
    (Sankyo Chemical Industries, Ltd.)
    Chair: Kunisuke Izawa (Ajinomoto)

  4. Scale-Up Engineering
    Madoka Kawasumi, Yasuo Hosono
    (Chiyoda Corporation)
    Chair: Koji Kagara

  5. Process Development of Amurubicin Hydrochloride (Anthracycline Anticancer Drug)
    Kazuhiko Takahashi
    (Sumitomo Chemical Co., Ltd. Organic Synthesus Research Laboratory)
    Chair: Toyonori Takebayashi (Sankyo)

  6. Selective Chemical Synthesis Using Microreactors
    Jun-ichi Yoshida
    (Department of Synthetic Chemistry and Biological Chemistry, Graduate aschool of Engineering, Kyoto University)
    Chair: Kiyoshi Tomioka (Kyoto Univ.)

  7. Development of a New Route toε-Caprolactam Precursor Using N-Hydroxyimide
    Satoshi Sakaguchi
    (Department of Applied Chemistry, Faculty of Engineering, Kansai University)
    Chair: Tatsuzo Ukita (Tanabe)

  8. Synthetic Studies on the Halichondrin B Analog, E7389
    Francis Gerard Fang
    iEisai Research Institutej
    Chair: Kuniaki Tatsuta (Waseda Univ.)

  9. Drug Development & Regulations---Recent Trends
    Ichiro Shinkai
    (Beta-Chem, Inc.)
    Chair: Toshiro Konoike (Shionogi)

<JSPC Award for Excellence 2004 Lecture>@Chair: Yoshihiro Matsumura (Nagasaki Univ.)

  1. Practical synthesis of 1b-methylcarbapenem utilizing a new dehydration Ti-Dieckmann condensation
    Ryohei Nagase, Naoki Manta, Tomonori Misaki, and Yoo Tanabe
    (Kwansei Gakuin Univ.)
    Makoto Sunagawa and Akira Sasaki
    (Sumitomo Pharmaceutical Co.)

  2. Resolution technology of racemic mixtures using distillation technique in industrial scale
    Yuuichi Katou, Tsutomu Sugawara, and Kazumi Okada
    (Nippon Kasei)

  3. Practical promotion system for carbonyl-ene reactions styrenes with paraformaldehyde - The combined use of boron trifluoride and molecular sieves
    Takahiro Okachi and Katsuhiko Fujimoto
    (Sankyo)

¡2005 JSPC Award for Excellence>>


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The Japanese Society for Process Chemistry